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-Structure paper
Title | Pharmacological Profile of BI 847325, an Orally Bioavailable, ATP-Competitive Inhibitor of MEK and Aurora Kinases. |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 15, Page 2388-2398, Year 2016 |
Publish date | Nov 25, 2015 (structure data deposition date) |
![]() | Sini, P. / Gurtler, U. / Zahn, S.K. / Baumann, C. / Rudolph, D. / Baumgartinger, R. / Strauss, E. / Haslinger, C. / Tontsch-Grunt, U. / Waizenegger, I.C. ...Sini, P. / Gurtler, U. / Zahn, S.K. / Baumann, C. / Rudolph, D. / Baumgartinger, R. / Strauss, E. / Haslinger, C. / Tontsch-Grunt, U. / Waizenegger, I.C. / Solca, F. / Bader, G. / Zoephel, A. / Treu, M. / Reiser, U. / Garin-Chesa, P. / Boehmelt, G. / Kraut, N. / Quant, J. / Adolf, G.R. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 2.7 Å |
Structure data | ![]() PDB-5eyk: ![]() PDB-5eym: ![]() PDB-5k3y: |
Chemicals | ![]() ChemComp-5U5: ![]() ChemComp-HOH: ![]() ChemComp-CA: ![]() ChemComp-6Q4: |
Source |
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![]() | TRANSFERASE / KINASE / Inhibitor |