+Search query
-Structure paper
Title | Mechanism of inhibition of human glucose transporter GLUT1 is conserved between cytochalasin B and phenylalanine amides. |
---|---|
Journal, issue, pages | Proc. Natl. Acad. Sci. USA, Vol. 113, Page 4711-4716, Year 2016 |
Publish date | Nov 12, 2015 (structure data deposition date) |
Authors | Kapoor, K. / Finer-Moore, J.S. / Pedersen, B.P. / Caboni, L. / Waight, A. / Hillig, R.C. / Bringmann, P. / Heisler, I. / Muller, T. / Siebeneicher, H. / Stroud, R.M. |
External links | Proc. Natl. Acad. Sci. USA / PubMed:27078104 |
Methods | X-ray diffraction |
Resolution | 2.9 - 3.002 Å |
Structure data | PDB-5eqg: PDB-5eqh: PDB-5eqi: |
Chemicals | ChemComp-5RE: ChemComp-5RF: ChemComp-5RH: |
Source |
|
Keywords | TRANSPORT PROTEIN/INHIBITOR / MFS transporter / glucose transporter / TRANSPORT PROTEIN-INHIBITOR complex |