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-Structure paper
Title | Crystal Structures of KPC-2 and SHV-1 beta-Lactamases in Complex with the Boronic Acid Transition State Analog S02030. |
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Journal, issue, pages | Antimicrob. Agents Chemother., Vol. 60, Page 1760-1766, Year 2016 |
Publish date | Oct 22, 2015 (structure data deposition date) |
![]() | Nguyen, N.Q. / Krishnan, N.P. / Rojas, L.J. / Prati, F. / Caselli, E. / Romagnoli, C. / Bonomo, R.A. / van den Akker, F. |
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Methods | X-ray diffraction |
Resolution | 1.54 - 1.87 Å |
Structure data | ![]() PDB-5ee8: ![]() PDB-5eec: |
Chemicals | ![]() ChemComp-ZXM: ![]() ChemComp-MA4: ![]() ChemComp-HOH: ![]() ChemComp-SO4: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / transition state inhibitor / HYDROLASE-HYDROLASE INHIBITOR complex |