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-Structure paper
Title | Structure-Guided Design of Group I Selective p21-Activated Kinase Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 5121-5136, Year 2015 |
Publish date | May 21, 2015 (structure data deposition date) |
![]() | Crawford, J.J. / Lee, W. / Aliagas, I. / Mathieu, S. / Hoeflich, K.P. / Zhou, W. / Wang, W. / Rouge, L. / Murray, L. / La, H. ...Crawford, J.J. / Lee, W. / Aliagas, I. / Mathieu, S. / Hoeflich, K.P. / Zhou, W. / Wang, W. / Rouge, L. / Murray, L. / La, H. / Liu, N. / Fan, P.W. / Cheong, J. / Heise, C.E. / Ramaswamy, S. / Mintzer, R. / Liu, Y. / Chao, Q. / Rudolph, J. |
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Methods | X-ray diffraction |
Resolution | 2.15 - 2.903 Å |
Structure data | ![]() PDB-4zy4: ![]() PDB-4zy5: ![]() PDB-4zy6: ![]() PDB-5bms: |
Chemicals | ![]() ChemComp-4T3: ![]() ChemComp-SO4: ![]() ChemComp-DMS: ![]() ChemComp-HOH: ![]() ChemComp-4T5: ![]() ChemComp-4T6: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / kinase / Inhibitor / Complex / TRANSFERASE-TRANSFERASE INHIBITOR complex / PAK1 |