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-Structure paper
Title | Exploiting Protein Conformational Change to Optimize Adenosine-Derived Inhibitors of Hsp70. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 4625-, Year 2016 |
Publish date | Sep 22, 2015 (structure data deposition date) |
Authors | Cheeseman, M.D. / Westwood, I.M. / Barbeau, O. / Rowlands, M.G. / Dobson, S. / Jones, A.M. / Jeganathan, F. / Burke, R. / Kadi, N. / Workman, P. ...Cheeseman, M.D. / Westwood, I.M. / Barbeau, O. / Rowlands, M.G. / Dobson, S. / Jones, A.M. / Jeganathan, F. / Burke, R. / Kadi, N. / Workman, P. / Collins, I. / Van Montfort, R.L.M. / Jones, K. |
External links | J. Med. Chem. / PubMed:27119979 |
Methods | X-ray diffraction |
Resolution | 1.65 - 1.9 Å |
Structure data | PDB-5aqz: PDB-5ar0: |
Chemicals | ChemComp-SGV: ChemComp-EDO: ChemComp-HOH: ChemComp-GB8: ChemComp-GOL: ChemComp-DMS: ChemComp-CL: |
Source |
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Keywords | CHAPERONE / HEAT SHOCK PROTEIN / HSP70 / HSP72 / ATPASE / ADENOSINE / INHIBITOR |