+Search query
-Structure paper
Title | Identification of an allosteric binding site for ROR gamma t inhibition. |
---|---|
Journal, issue, pages | Nat Commun, Vol. 6, Page 8833-8833, Year 2015 |
Publish date | Mar 13, 2015 (structure data deposition date) |
![]() | Scheepstra, M. / Leysen, S. / van Almen, G.C. / Miller, J.R. / Piesvaux, J. / Kutilek, V. / van Eenennaam, H. / Zhang, H. / Barr, K. / Nagpal, S. ...Scheepstra, M. / Leysen, S. / van Almen, G.C. / Miller, J.R. / Piesvaux, J. / Kutilek, V. / van Eenennaam, H. / Zhang, H. / Barr, K. / Nagpal, S. / Soisson, S.M. / Kornienko, M. / Wiley, K. / Elsen, N. / Sharma, S. / Correll, C.C. / Trotter, B.W. / van der Stelt, M. / Oubrie, A. / Ottmann, C. / Parthasarathy, G. / Brunsveld, L. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.77 - 2.32 Å |
Structure data | ![]() PDB-4ypq: ![]() PDB-5c4o: ![]() PDB-5c4s: ![]() PDB-5c4t: ![]() PDB-5c4u: |
Chemicals | ![]() ChemComp-4F1: ![]() ChemComp-MG: ![]() ChemComp-HOH: ![]() ChemComp-GOL: ![]() ChemComp-SO4: ![]() ChemComp-4Y5: ![]() ChemComp-4Y6: ![]() ChemComp-4Y7: |
Source |
|
![]() | TRANSCRIPTION / nuclear receptor ligand binding domain / TRANSCRIPTION/TRANSCRIPTION INHIBITOR / Allosteric / Inhibitor / TRANSCRIPTION-TRANSCRIPTION INHIBITOR complex |