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-Structure paper
Title | Structural Insights Into Fgfr Kinase Isoform Selectivity: Diverse Binding Modes of Azd4547 and Ponatinib in Complex with Fgfr1 and Fgfr4 |
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Journal, issue, pages | Structure, Vol. 22, Page 1764-, Year 2014 |
Publish date | Aug 27, 2014 (structure data deposition date) |
![]() | Tucker, J.A. / Klein, T. / Breed, J. / Breeze, A.L. / Overman, R. / Phillips, C. / Norman, R.A. |
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Methods | X-ray diffraction |
Resolution | 1.85 - 2.57 Å |
Structure data | ![]() PDB-4uxq: ![]() PDB-4v01: ![]() PDB-4v04: ![]() PDB-4v05: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-0LI: ![]() ChemComp-HOH: ![]() ChemComp-EDO: ![]() ChemComp-66T: |
Source |
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![]() | TRANSFERASE / KINASE DFG-OUT FGFR INHIBITOR COMPLEX |