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-Structure paper
Title | Human Sterol 14Alpha-Demethylase (Cyp51) as a Target for Anticancer Chemotherapy: Towards Structure-Aided Drug Design. |
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Journal, issue, pages | J. Lipid Res., Vol. 57, Page 1552-, Year 2016 |
Publish date | Mar 24, 2015 (structure data deposition date) |
![]() | Hargrove, T.Y. / Friggeri, L. / Wawrzak, Z. / Sivakumaran, S. / Yazlovitskaya, E.M. / Hiebert, S.W. / Guengerich, F.P. / Waterman, M.R. / Lepesheva, G.I. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.04 - 2.5 Å |
Structure data | ![]() PDB-4uhi: ![]() PDB-4uhl: |
Chemicals | ![]() ChemComp-HEM: ![]() ChemComp-VFV: ![]() ChemComp-HOH: |
Source |
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![]() | OXIDOREDUCTASE / MONOOXYGENASE / STEROL BIOSYNTHESIS / EUKARYOTIC MEMBRANES / CYTOCHROME P450 FOLD / ENDOPLASMIC RETICULUM / CYTOCHROME P450 / CYP51 |