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-Structure paper
Title | Covalent docking of large libraries for the discovery of chemical probes. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 10, Page 1066-1072, Year 2014 |
Publish date | Jul 25, 2013 (structure data deposition date) |
![]() | London, N. / Miller, R.M. / Krishnan, S. / Uchida, K. / Irwin, J.J. / Eidam, O. / Gibold, L. / Cimermancic, P. / Bonnet, R. / Shoichet, B.K. / Taunton, J. |
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Methods | X-ray diffraction |
Resolution | 1.42 - 3 Å |
Structure data | ![]() PDB-4lv0: ![]() PDB-4lv1: ![]() PDB-4lv2: ![]() PDB-4lv3: ![]() PDB-4m8t: |
Chemicals | ![]() ChemComp-APB: ![]() ChemComp-PO4: ![]() ChemComp-HOH: ![]() ChemComp-NL9: ![]() ChemComp-N95: ![]() ChemComp-25N: ![]() ChemComp-RMM: ![]() ChemComp-NA: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / AMPC BETA-LACTAMASE / CLASS C / HYDROLASE / BORONIC ACID / COVALENT INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex / TRANSFERASE/TRANSFERASE INHIBITOR / Protein Kinase / Phosphorylation / TRANSFERASE-TRANSFERASE INHIBITOR complex |