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-Structure paper
Title | Thermodynamic and structural analysis of HIV protease resistance to darunavir - analysis of heavily mutated patient-derived HIV-1 proteases. |
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Journal, issue, pages | Febs J., Vol. 281, Page 1834-1847, Year 2014 |
Publish date | Sep 15, 2011 (structure data deposition date) |
![]() | Kozisek, M. / Lepsik, M. / Grantz Saskova, K. / Brynda, J. / Konvalinka, J. / Rezacova, P. |
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Methods | X-ray diffraction |
Resolution | 1.95 - 2.23 Å |
Structure data | ![]() PDB-3ttp: ![]() PDB-4ll3: |
Chemicals | ![]() ChemComp-017: ![]() ChemComp-CL: ![]() ChemComp-BME: ![]() ChemComp-HOH: |
Source |
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![]() | Hydrolase/hydrolase inhibitor / hydrolase / viral praticle / Hydrolase-hydrolase inhibitor complex / Hydrolase Inhibitor-darunavir / HIV-1 protease / TMC114 |