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-Structure paper
Title | 4-Phenyl-7-Azaindoles as Potent, Selective and Bioavailable Ikk2 Inhibitors Demonstrating Good in Vivo Efficacy. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 22, Page 5222-, Year 2012 |
Publish date | Jun 3, 2012 (structure data deposition date) |
![]() | Liddle, J. / Bamborough, P. / Barker, M.D. / Campos, S. / Chung, C. / Cousins, R.P.C. / Faulder, P. / Heathcote, M.L. / Hobbs, H. / Holmes, D.S. ...Liddle, J. / Bamborough, P. / Barker, M.D. / Campos, S. / Chung, C. / Cousins, R.P.C. / Faulder, P. / Heathcote, M.L. / Hobbs, H. / Holmes, D.S. / Ioannou, C. / Ramirez-Molina, C. / Morse, M.A. / Osborn, R. / Payne, J.J. / Pritchard, J.M. / Rumsey, W.L. / Tape, D.T. / Vicentini, G. / Whitworth, C. / Williamson, R.A. |
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Methods | X-ray diffraction |
Resolution | 1.91 Å |
Structure data | ![]() PDB-4awi: |
Chemicals | ![]() ChemComp-AQ2: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE |