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-Structure paper
Title | X-ray structures of progesterone receptor ligand binding domain in its agonist state reveal differing mechanisms for mixed profiles of 11 beta-substituted steroids. |
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Journal, issue, pages | J. Biol. Chem., Vol. 287, Page 20333-20343, Year 2012 |
Publish date | Sep 27, 2011 (structure data deposition date) |
![]() | Lusher, S.J. / Raaijmakers, H.C. / Vu-Pham, D. / Kazemier, B. / Bosch, R. / McGuire, R. / Azevedo, R. / Hamersma, H. / Dechering, K. / Oubrie, A. ...Lusher, S.J. / Raaijmakers, H.C. / Vu-Pham, D. / Kazemier, B. / Bosch, R. / McGuire, R. / Azevedo, R. / Hamersma, H. / Dechering, K. / Oubrie, A. / van Duin, M. / de Vlieg, J. |
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Methods | X-ray diffraction |
Resolution | 1.9 - 2 Å |
Structure data | ![]() PDB-4a2j: ![]() PDB-4apu: |
Chemicals | ![]() ChemComp-AS0: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-OR8: ![]() ChemComp-A2K: |
Source |
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![]() | TRANSCRIPTION / PARTIAL AGONIST / ASOPRISNIL |