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-Structure paper
Title | Structure-Based Library Design and the Discovery of a Potent and Selective Mast Cell Beta-Tryptase Inhibitor as an Oral Therapeutic Agent. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 22, Page 1049-, Year 2012 |
Publish date | Nov 4, 2011 (structure data deposition date) |
![]() | Liang, G. / Aldous, S. / Merriman, G. / Levell, J. / Pribish, J. / Cairns, J. / Chen, X. / Maignan, S. / Mathieu, M. / Tsay, J. ...Liang, G. / Aldous, S. / Merriman, G. / Levell, J. / Pribish, J. / Cairns, J. / Chen, X. / Maignan, S. / Mathieu, M. / Tsay, J. / Sides, K. / Rebello, S. / Whitely, B. / Morize, I. / Pauls, H.W. |
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Methods | X-ray diffraction |
Resolution | 2.05 Å |
Structure data | ![]() PDB-4a6l: |
Chemicals | ![]() ChemComp-P43: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / INHIBITOR |