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-Structure paper
Title | EC144 Is a Potent Inhibitor of the Heat Shock Protein 90. |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 7786-7795, Year 2012 |
Publish date | Jan 18, 2011 (structure data deposition date) |
Authors | Shi, J. / Van de Water, R. / Hong, K. / Lamer, R.B. / Weichert, K.W. / Sandoval, C.M. / Kasibhatla, S.R. / Boehm, M.F. / Chao, J. / Lundgren, K. ...Shi, J. / Van de Water, R. / Hong, K. / Lamer, R.B. / Weichert, K.W. / Sandoval, C.M. / Kasibhatla, S.R. / Boehm, M.F. / Chao, J. / Lundgren, K. / Timple, N. / Lough, R. / Ibanez, G. / Boykin, C. / Burrows, F.J. / Kehry, M.R. / Yun, T.J. / Harning, E.K. / Ambrose, C. / Thompson, J. / Bixler, S.A. / Dunah, A. / Snodgrass-Belt, P. / Arndt, J. / Enyedy, I.J. / Li, P. / Hong, V.S. / McKenzie, A. / Biamonte, M.A. |
External links | J. Med. Chem. / PubMed:22938030 |
Methods | X-ray diffraction |
Resolution | 1.79 Å |
Structure data | PDB-3qdd: |
Chemicals | ChemComp-94M: ChemComp-HOH: |
Source |
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Keywords | CHAPERONE/CHAPERONE INHIBITOR / ATPase / CHAPERONE-CHAPERONE INHIBITOR complex |