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-Structure paper
Title | Structure based evolution of a novel series of positive modulators of the AMPA receptor. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 21, Page 805-811, Year 2011 |
Publish date | Nov 18, 2010 (structure data deposition date) |
Authors | Jamieson, C. / Maclean, J.K. / Brown, C.I. / Campbell, R.A. / Gillen, K.J. / Gillespie, J. / Kazemier, B. / Kiczun, M. / Lamont, Y. / Lyons, A.J. ...Jamieson, C. / Maclean, J.K. / Brown, C.I. / Campbell, R.A. / Gillen, K.J. / Gillespie, J. / Kazemier, B. / Kiczun, M. / Lamont, Y. / Lyons, A.J. / Moir, E.M. / Morrow, J.A. / Pantling, J. / Rankovic, Z. / Smith, L. |
External links | Bioorg. Med. Chem. Lett. / PubMed:21190850 |
Methods | X-ray diffraction |
Resolution | 1.8 - 2.2 Å |
Structure data | PDB-3pmv: PDB-3pmw: PDB-3pmx: |
Chemicals | ChemComp-GLU: ChemComp-SO4: ChemComp-557: ChemComp-GOL: ChemComp-HOH: ChemComp-DMS: ChemComp-G69: ChemComp-EDO: ChemComp-808: |
Source |
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Keywords | TRANSPORT PROTEIN / Membrane protein / Fusion protein / chimera protein |