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Structure paper

TitleQuinolines as a novel structural class of potent and selective PDE4 inhibitors. Optimisation for inhaled administration.
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 19, Page 5261-5265, Year 2009
Publish dateApr 1, 2009 (structure data deposition date)
AuthorsWoodrow, M.D. / Ballantine, S.P. / Barker, M.D. / Clarke, B.J. / Dawson, J. / Dean, T.W. / Delves, C.J. / Evans, B. / Gough, S.L. / Guntrip, S.B. ...Woodrow, M.D. / Ballantine, S.P. / Barker, M.D. / Clarke, B.J. / Dawson, J. / Dean, T.W. / Delves, C.J. / Evans, B. / Gough, S.L. / Guntrip, S.B. / Holman, S. / Holmes, D.S. / Kranz, M. / Lindvaal, M.K. / Lucas, F.S. / Neu, M. / Ranshaw, L.E. / Solanke, Y.E. / Somers, D.O. / Ward, P. / Wiseman, J.O.
External linksBioorg. Med. Chem. Lett. / PubMed:19656678
MethodsX-ray diffraction
Resolution1.75 Å
Structure data

PDB-3gwt:
Catalytic domain of human phosphodiesterase 4B2B in complex with a quinoline inhibitor
Method: X-RAY DIFFRACTION / Resolution: 1.75 Å

Chemicals

ChemComp-066:
6-{[3-(dimethylcarbamoyl)phenyl]sulfonyl}-4-[(3-methoxyphenyl)amino]-8-methylquinoline-3-carboxamide

ChemComp-ZN:
Unknown entry

ChemComp-MG:
Unknown entry

ChemComp-ARS:
ARSENIC

ChemComp-GOL:
GLYCEROL

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsHYDROLASE / PDE / PHOSPHODIESTERASE / cAMP

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