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-Structure paper
Title | Structure of a small-molecule inhibitor of a DNA polymerase sliding clamp. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. Usa, Vol. 105, Page 11116-11121, Year 2008 |
Publish date | May 5, 2008 (structure data deposition date) |
![]() | Georgescu, R.E. / Yurieva, O. / Kim, S.S. / Kuriyan, J. / Kong, X.P. / O'Donnell, M. |
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Methods | X-ray diffraction |
Resolution | 1.64 - 2 Å |
Structure data | ![]() PDB-3d1e: ![]() PDB-3d1f: ![]() PDB-3d1g: |
Chemicals | ![]() ChemComp-HOH: ![]() ChemComp-PEG: ![]() ChemComp-323: ![]() ChemComp-322: |
Source |
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![]() | TRANSFERASE / TRANSCRIPTION / chemical probe / DNA polymerase / DNA sliding clamp / DNA replication / rational drug design / antibiotic target |