+Search query
-Structure paper
Title | Structural basis for binding of cyclic 2-oxoglutarate analogues to factor-inhibiting hypoxia-inducible factor. |
---|---|
Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 20, Page 6125-6128, Year 2010 |
Publish date | Oct 10, 2008 (structure data deposition date) |
![]() | Conejo-Garcia, A. / McDonough, M.A. / Loenarz, C. / McNeill, L.A. / Hewitson, K.S. / Ge, W. / Lienard, B.M. / Schofield, C.J. / Clifton, I.J. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.12 - 2.5 Å |
Structure data | ![]() PDB-2w0x: ![]() PDB-2wa3: ![]() PDB-2wa4: |
Chemicals | ![]() ChemComp-FE2: ![]() ChemComp-PD2: ![]() ChemComp-SO4: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-A29: ![]() ChemComp-069: |
Source |
|
![]() | OXIDOREDUCTASE / HYDROXYLASE / DIOXYGENASE / TRANSCRIPTION / TRANSCRIPTION ACTIVATOR/INHIBITOR / HYPOXIA |