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Title | Crystal Structures for HIV-1 Reverse Transcriptase in Complexes with Three Pyridinone Derivatives: A New Class of Non-Nucleoside Inhibitors Effective against a Broad Range of Drug-Resistant Strains. |
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Journal, issue, pages | J. Med. Chem., Vol. 48, Page 7582-7591, Year 2005 |
Publish date | Sep 28, 2005 (structure data deposition date) |
Authors | Himmel, D.M. / Das, K. / Clark Jr., A.D. / Hughes, S.H. / Benjahad, A. / Oumouch, S. / Guillemont, J. / Coupa, S. / Poncelet, A. / Csoka, I. ...Himmel, D.M. / Das, K. / Clark Jr., A.D. / Hughes, S.H. / Benjahad, A. / Oumouch, S. / Guillemont, J. / Coupa, S. / Poncelet, A. / Csoka, I. / Meyer, C. / Andries, K. / Nguyen, C.H. / Grierson, D.S. / Arnold, E. |
External links | J. Med. Chem. / PubMed:16302798 |
Methods | X-ray diffraction |
Resolution | 2.43 - 2.95 Å |
Structure data | PDB-2b5j: PDB-2ban: PDB-2be2: |
Chemicals | ChemComp-MN: ChemComp-3AC: ChemComp-HOH: ChemComp-357: ChemComp-GOL: ChemComp-R22: |
Source |
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Keywords | TRANSFERASE / AIDS / HIV / DRUG DESIGN / REVERSE TRANSCRIPTASE / RT / PROTEIN-INHIBITOR COMPLEX / DRUG RESISTANCE |