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TitleImidazo[1,2-A]Pyridines: A Potent and Selective Class of Cyclin-Dependent Kinase Inhibitors Identified Through Structure-Based Hybridisation
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 13, Page 3021-, Year 2003
Publish dateJun 24, 2003 (structure data deposition date)
AuthorsAnderson, M. / Beattie, J.F. / Breault, G.A. / Breed, J. / Byth, K.F. / Culshaw, J.D. / Ellston, R.P.A. / Green, S. / Minshull, C.A. / Norman, R.A. ...Anderson, M. / Beattie, J.F. / Breault, G.A. / Breed, J. / Byth, K.F. / Culshaw, J.D. / Ellston, R.P.A. / Green, S. / Minshull, C.A. / Norman, R.A. / Pauptit, R.A. / Stanway, J. / Thomas, A.P. / Jewsbury, P.J.
External linksBioorg. Med. Chem. Lett. / PubMed:12941325
MethodsX-ray diffraction
Resolution1.6 - 2.31 Å
Structure data

PDB-1oiq:
Imidazopyridines: a potent and selective class of Cyclin-dependent Kinase inhibitors identified through Structure-based hybridisation
Method: X-RAY DIFFRACTION / Resolution: 2.31 Å

PDB-1oir:
Imidazopyridines: a potent and selective class of Cyclin-dependent Kinase inhibitors identified through Structure-based hybridisation
Method: X-RAY DIFFRACTION / Resolution: 1.91 Å

PDB-1oit:
Imidazopyridines: a potent and selective class of Cyclin-dependent Kinase inhibitors identified through Structure-based hybridisation
Method: X-RAY DIFFRACTION / Resolution: 1.6 Å

Chemicals

ChemComp-HDU:
N-[4-(2-METHYLIMIDAZO[1,2-A]PYRIDIN-3-YL)-2-PYRIMIDINYL]ACETAMIDE

ChemComp-HOH:
WATER

ChemComp-HDY:
1-(DIMETHYLAMINO)-3-(4-{{4-(2-METHYLIMIDAZO[1,2-A]PYRIDIN-3-YL)PYRIMIDIN-2-YL]AMINO}PHENOXY)PROPAN-2-OL

ChemComp-HDT:
4-[(4-IMIDAZO[1,2-A]PYRIDIN-3-YLPYRIMIDIN-2-YL)AMINO]BENZENESULFONAMIDE

Source
  • homo sapiens (human)
KeywordsKINASE / PROTEIN KINASE / TRANSFERASE / SERINE/THREONINE-PROTEIN KINASE / ATP-BINDING / CELL CYCLE / CELL DIVISION / MITOSIS / PHOSPHORYLATION

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