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-Structure paper
Title | Unexpected formation of an epoxide-derived multisubstrate adduct inhibitor on the active site of GAR transformylase. |
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Journal, issue, pages | Biochemistry, Vol. 40, Page 13538-13547, Year 2001 |
Publish date | Jul 13, 2001 (structure data deposition date) |
Authors | Greasley, S.E. / Marsilje, T.H. / Cai, H. / Baker, S. / Benkovic, S.J. / Boger, D.L. / Wilson, I.A. |
External links | Biochemistry / PubMed:11695901 |
Methods | X-ray diffraction |
Resolution | 1.6 Å |
Structure data | PDB-1jkx: |
Chemicals | ChemComp-138: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / PURINE BIOSYNTHESIS / ANTI-CANCER AGENT / ENZYME-ASSEMBLED MULTISUBSTRATE ADDUCT INHIBITOR COMPLEX |