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-Structure paper
| Title | Molecular Glue Prodrug Discovery Enabled by Targeted Degron Display |
|---|---|
| Journal, issue, pages | To Be Published |
| Publish date | Jun 27, 2025 (structure data deposition date) |
Authors | Zhuang Z / Woong Sub B / Chrustowicz J / Kozicka Z / Hinshaw SM / Li VL / Donovan KA / Sepic S / You I / Slabicki M ...Zhuang Z / Woong Sub B / Chrustowicz J / Kozicka Z / Hinshaw SM / Li VL / Donovan KA / Sepic S / You I / Slabicki M / Fischer ES / Ebert BL / Schulman BA / Gray NS |
External links | Search PubMed |
| Methods | EM (single particle) |
| Resolution | 3.38 - 11.77 Å |
| Structure data | ![]() EMDB-54194: ZZ1-SO2H-induced assembly of the YPEL5-CTLH E3 ligase and BRD4(BD1) neosubstrate EMDB-54215, PDB-9rsc: EMDB-54216, PDB-9rsd: |
| Chemicals | ![]() ChemComp-ZN: ![]() PDB-1il8: ![]() ChemComp-HOH: ![]() PDB-1il9: |
| Source |
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Keywords | LIGASE / E3 ubiquitin ligase / CTLH / GID / YPEL5 / Molecular Glue Degrader / Targeted Protein Degradation |
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homo sapiens (human)
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