タイトル Fragment-based drug discovery for transthyretin kinetic stabilisers using a novel capillary zone electrophoresis method. ジャーナル・号・ページ Plos One , Vol. 20, Page e0323816-e0323816, Year 2025掲載日 2024年10月27日 (構造データの登録日) 著者Chen, W. リンク Plos One / PubMed:40367241手法 X線回折 解像度 1.18 - 1.76 Å 構造データ PDB-9h7a : 構造ビューア Human Transthyretin in Complex with 3,5-Dichlorobenzenesulfonamide 手法 : X-RAY DIFFRACTION / 解像度 : 1.76 Å
PDB-9h7b : 構造ビューア Human Transthyretin in Complex with Biphenyl-4-carboxylic Acid手法 : X-RAY DIFFRACTION / 解像度 : 1.51 Å
PDB-9h7c : 構造ビューア Human Transthyretin in Complex with 4-(1H-imidazol-1-yl)phenol 手法 : X-RAY DIFFRACTION / 解像度 : 1.27 Å
PDB-9h7d : 構造ビューア Human Transthyretin in Complex with 2-(phenylamino)benzoic acid手法 : X-RAY DIFFRACTION / 解像度 : 1.23 Å
PDB-9h7e : 構造ビューア Human Transthyretin in Complex with 4-pyridin-3-ylbenzoic acid手法 : X-RAY DIFFRACTION / 解像度 : 1.43 Å
PDB-9h7f : 構造ビューア Human Transthyretin in Complex with 3,5-dichloroaniline 手法 : X-RAY DIFFRACTION / 解像度 : 1.24 Å
PDB-9h7g : 構造ビューア Human Transthyretin in Complex with 1H-indole-3-carbonitrile 手法 : X-RAY DIFFRACTION / 解像度 : 1.49 Å
PDB-9h7h : 構造ビューア Human Transthyretin in Complex with Isoquinolin-3-amine 手法 : X-RAY DIFFRACTION / 解像度 : 1.47 Å
PDB-9h7i : 構造ビューア Human Transthyretin in Complex with 4-(1H-pyrazol-4-yl)quinoline 手法 : X-RAY DIFFRACTION / 解像度 : 1.21 Å
PDB-9h7j : 構造ビューア Human Transthyretin in Complex with 5-methyl-4-phenyl-1H-pyrazol-3-amine 手法 : X-RAY DIFFRACTION / 解像度 : 1.3 Å
PDB-9h7k : 構造ビューア Human Transthyretin in Complex with 8-(3,5-dimethyl-1H-pyrazol-4-yl)quinoline 手法 : X-RAY DIFFRACTION / 解像度 : 1.6 Å
PDB-9h7l : 構造ビューア Human Transthyretin in Complex with 4-phenyl-1H-pyrazolo[3,4-b]pyridin-3-amine 手法 : X-RAY DIFFRACTION / 解像度 : 1.18 Å
PDB-9h7m : 構造ビューア Human Transthyretin in Complex with 4-(quinolin-8-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine 手法 : X-RAY DIFFRACTION / 解像度 : 1.27 Å
PDB-9h7n : 構造ビューア Human Transthyretin in Complex with 4-(5-methyl-1H-1,2,4-triazol-3-yl)quinoline 手法 : X-RAY DIFFRACTION / 解像度 : 1.26 Å
PDB-9h7o : 構造ビューア Human Transthyretin in Complex with 5-(quinolin-8-yl)pyrimidin-2-amine 手法 : X-RAY DIFFRACTION / 解像度 : 1.24 Å
PDB-9h7p : 構造ビューア Human Transthyretin S52P Mutant in Complex with 4-(1H-pyrazol-4-yl)quinoline手法 : X-RAY DIFFRACTION / 解像度 : 1.36 Å
化合物 PDB-1isu : 構造ビューア THE THREE-DIMENSIONAL STRUCTURE OF THE HIGH-POTENTIAL IRON-SULFUR PROTEIN ISOLATED FROM THE PURPLE PHOTOTROPHIC BACTERIUM RHODOCYCLUS TENUIS DETERMINED AND REFINED AT 1.5 ANGSTROMS RESOLUTION
PDB-1iss : 構造ビューア Crystal Structure of Metabotropic Glutamate Receptor Subtype 1 Complexed with an antagonist
PDB-1isy : 構造ビューア Crystal structure of xylanase from Streptomyces olivaceoviridis E-86 complexed with glucose
PDB-1is2 : 構造ビューア Crystal Structure of Peroxisomal Acyl-CoA Oxidase-II from Rat Liver
PDB-1is0 : 構造ビューア Crystal Structure of a Complex of the Src SH2 Domain with Conformationally Constrained Peptide Inhibitor
PDB-1isv : 構造ビューア Crystal structure of xylanase from Streptomyces olivaceoviridis E-86 complexed with xylose
PDB-1ist : 構造ビューア Crystal structure of yeast cyclophilin A, CPR1
PDB-1isz : 構造ビューア Crystal structure of xylanase from Streptomyces olivaceoviridis E-86 complexed with galactose
由来 homo sapiens (ヒト) キーワード TRANSPORT PROTEIN / Amyloidosis / Retinol / Thyroxine / RBP