タイトル | Diverse Human Therapeutics Impact Hormone and Neurotransmitter Homeostasis by Inhibiting Gut Microbial Enzymes |
---|
ジャーナル・号・ページ | To Be Published |
---|
掲載日 | 2023年3月7日 (構造データの登録日) |
---|
著者 | Simpson, J.B. / Redinbo, M.R. |
---|
リンク | PubMedで検索 |
---|
手法 | X線回折 |
---|
解像度 | 2.4 - 2.94 Å |
---|
構造データ | PDB-8gen: E. eligens beta-glucuronidase bound to UNC10201652-glucuronide 手法: X-RAY DIFFRACTION / 解像度: 2.94 Å PDB-8geo: E. eligens beta-glucuronidase bound to 3-OH-desloratidine-glucuronide 手法: X-RAY DIFFRACTION / 解像度: 2.89 Å PDB-8geq: E. eligens beta-glucuronidase bound to ceritinib-glucuronide 手法: X-RAY DIFFRACTION / 解像度: 2.75 Å PDB-8ger: E. eligens beta-glucuronidase bound to norquetiapine-glucuronide 手法: X-RAY DIFFRACTION / 解像度: 2.4 Å PDB-8ges: R. hominis 2 beta-glucuronidase bound to UNC10201652-glucuronide 手法: X-RAY DIFFRACTION / 解像度: 2.7 Å PDB-8get: R. hominis 2 beta-glucuronidase bound to norquetiapine-glucuronide 手法: X-RAY DIFFRACTION / 解像度: 2.9 Å |
---|
化合物 | ChemComp-I9G: 8-(4-beta-D-glucopyranuronosylpiperazin-1-yl)-5-(morpholin-4-yl)-1,2,3,4-tetrahydro[1,2,3]triazino[4',5':4,5]thieno[2,3
|
---|
由来 | - lachnospira eligens (バクテリア)
- roseburia hominis (バクテリア)
|
---|
キーワード | HYDROLASE / beta-glucuronidase / inhibitor / glucuronide |
---|