タイトル | Structure of the BCL6 BTB domain |
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ジャーナル・号・ページ | To Be Published |
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掲載日 | 2021年8月18日 (構造データの登録日) |
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著者 | Watson, I. / Isaac, M. |
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リンク | PubMedで検索 |
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手法 | X線回折 |
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解像度 | 1.25 - 2.21 Å |
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構造データ | PDB-7rv3: Crystal structure of the BCL6 BTB domain in complex with OICR-9124 手法: X-RAY DIFFRACTION / 解像度: 1.35 Å PDB-7rv4: Crystal structure of the BCL6 BTB domain in complex with OICR-9153 手法: X-RAY DIFFRACTION / 解像度: 1.25 Å PDB-7rv5: Crystal structure of the BCL6 BTB domain in complex with OICR-9287 手法: X-RAY DIFFRACTION / 解像度: 2.21 Å PDB-7rv6: Crystal structure of the BCL6 BTB domain in complex with OICR-9288 手法: X-RAY DIFFRACTION / 解像度: 1.683 Å PDB-7rv7: Crystal structure of the BCL6 BTB domain in complex with OICR-9322 手法: X-RAY DIFFRACTION / 解像度: 1.63 Å PDB-7rv8: Crystal structure of the BCL6 BTB domain in complex with OICR-10268 手法: X-RAY DIFFRACTION / 解像度: 1.25 Å PDB-7rv9: Crystal structure of the BCL6 BTB domain in complex with OICR-10269 手法: X-RAY DIFFRACTION / 解像度: 1.5 Å |
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化合物 | ChemComp-7R5: N-(3-chloropyridin-4-yl)-2-[2-(morpholin-4-yl)-4-oxo-3,4-dihydro-7H-pyrrolo[2,3-d]pyrimidin-7-yl]acetamide
ChemComp-7SO: N-(3-chloropyridin-4-yl)-2-{5-(3-cyanophenyl)-3-[3-(1-methyl-1H-pyrazol-4-yl)prop-2-yn-1-yl]-4-oxo-3,4-dihydro-7H-pyrrolo[2,3-d]pyrimidin-7-yl}acetamide
ChemComp-7RB: 2-[2-(4-benzylpiperidin-1-yl)-4-oxo-3,4-dihydro-7H-pyrrolo[2,3-d]pyrimidin-7-yl]-N-(3-chloropyridin-4-yl)acetamide
ChemComp-7SC: N-(3-chloropyridin-4-yl)-2-{4-oxo-2-[(2-phenylethyl)amino]-3,4-dihydro-7H-pyrrolo[2,3-d]pyrimidin-7-yl}acetamide
ChemComp-7SH: N-(3-chloropyridin-4-yl)-2-{5-(3-cyano-4-hydroxyphenyl)-3-[3-(1-methyl-1H-pyrazol-4-yl)prop-2-yn-1-yl]-4-oxo-3,4-dihydro-7H-pyrrolo[2,3-d]pyrimidin-7-yl}acetamide
ChemComp-7ST: N-[5-chloro-2-(morpholin-4-yl)pyridin-4-yl]-2-{5-(3-cyano-4-hydroxy-5-methylphenyl)-3-[3-(1-methyl-1H-pyrazol-4-yl)prop-2-yn-1-yl]-4-oxo-3,4-dihydro-7H-pyrrolo[2,3-d]pyrimidin-7-yl}acetamide
ChemComp-7SZ: N-[5-chloro-2-(4-methylpiperazin-1-yl)pyridin-4-yl]-2-{5-(3-cyano-4-hydroxy-5-methylphenyl)-3-[3-(1-methyl-1H-pyrazol-4-yl)prop-2-yn-1-yl]-4-oxo-3,4-dihydro-7H-pyrrolo[2,3-d]pyrimidin-7-yl}acetamide
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由来 | - homo sapiens (ヒト)
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キーワード | TRANSCRIPTION / immunity / inflammatory response / transcription repressor |
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