Screening of a Custom-Designed Acid Fragment Library Identifies 1-Phenylpyrroles and 1-Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity.
PDB-6ysk: 1-phenylpyrroles and 1-enylpyrrolidines as inhibitors of Notum 手法: X-RAY DIFFRACTION / 解像度: 1.21 Å
PDB-6yuw: STRUCTURE OF THE WNT DEACYLASE NOTUM IN COMPLEX WITH A PYRROLE-3-CARBOXYLIC ACID FRAGMENT 454 手法: X-RAY DIFFRACTION / 解像度: 1.94 Å
PDB-6yuy: STRUCTURE OF THE WNT DEACYLASE NOTUM IN COMPLEX WITH A PYRROLE-3-CARBOXYLIC ACID FRAGMENT 471 手法: X-RAY DIFFRACTION / 解像度: 2.0 Å
PDB-6yv0: STRUCTURE OF THE WNT DEACYLASE NOTUM IN COMPLEX WITH A PYRROLIDINE-3-CARBOXYLIC ACID FRAGMENT 587 手法: X-RAY DIFFRACTION / 解像度: 2.0 Å
PDB-6yv2: STRUCTURE OF THE WNT DEACYLASE NOTUM IN COMPLEX WITH A PYRROLIDINE-3-CARBOXYLIC ACID FRAGMENT 598 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å
PDB-6yv4: STRUCTURE OF THE WNT DEACYLASE NOTUM IN COMPLEX WITH A PYRROLE-3-CARBOXYLIC ACID FRAGMENT 686 手法: X-RAY DIFFRACTION / 解像度: 2.0 Å
PDB-6yxi: Structure of Notum in complex with a 1-(3-Chlorophenyl)-2,5-dimethyl-1H-pyrrole-3-carboxylic acid inhibitor 手法: X-RAY DIFFRACTION / 解像度: 1.34 Å