タイトル | Kinase Scaffold Repurposing in the Public Domain |
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ジャーナル・号・ページ | To be published |
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掲載日 | 2019年6月18日 (構造データの登録日) |
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著者 | Sorrell, F.J. / Henderson, S.H. / Elkins, J.M. / Ward, S. |
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リンク | PubMedで検索 |
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手法 | X線回折 |
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解像度 | 1.05 - 2.445 Å |
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構造データ | PDB-6s11: Crystal Structure of DYRK1A with small molecule inhibitor 手法: X-RAY DIFFRACTION / 解像度: 2.445 Å PDB-6s14: Crystal Structure of DYRK1A with small molecule inhibitor 手法: X-RAY DIFFRACTION / 解像度: 1.05 Å PDB-6s17: Crystal Structure of DYRK1A with small molecule inhibitor 手法: X-RAY DIFFRACTION / 解像度: 1.1 Å PDB-6s1b: Crystal Structure of DYRK1A with small molecule inhibitor 手法: X-RAY DIFFRACTION / 解像度: 1.3 Å PDB-6s1h: Crystal Structure of DYRK1A with small molecule inhibitor 手法: X-RAY DIFFRACTION / 解像度: 1.05 Å PDB-6s1j: Crystal Structure of DYRK1A with small molecule inhibitor 手法: X-RAY DIFFRACTION / 解像度: 1.408 Å |
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化合物 | ChemComp-KQE: 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine
ChemComp-KQW: ~{N}-cyclopropyl-~{N}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine
ChemComp-KQK: ~{N},~{N}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine
ChemComp-KRQ: ~{N}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine
ChemComp-KQZ: ~{N},~{N}-dimethyl-4-(1~{H}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine
ChemComp-KRK: 3-[2-[(3~{S})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazine
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由来 | - homo sapiens (ヒト)
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キーワード | TRANSFERASE / Kinase / catalytic domain / phosphorylated |
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