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-Structure paper
タイトル | Discovery and Optimization of a Selective Ligand for the Switch/Sucrose Nonfermenting-Related Bromodomains of Polybromo Protein-1 by the Use of Virtual Screening and Hydration Analysis. |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 59, Page 8787-8803, Year 2016 |
掲載日 | 2016年1月24日 (構造データの登録日) |
![]() | Myrianthopoulos, V. / Gaboriaud-Kolar, N. / Tallant, C. / Hall, M.L. / Grigoriou, S. / Brownlee, P.M. / Fedorov, O. / Rogers, C. / Heidenreich, D. / Wanior, M. ...Myrianthopoulos, V. / Gaboriaud-Kolar, N. / Tallant, C. / Hall, M.L. / Grigoriou, S. / Brownlee, P.M. / Fedorov, O. / Rogers, C. / Heidenreich, D. / Wanior, M. / Drosos, N. / Mexia, N. / Savitsky, P. / Bagratuni, T. / Kastritis, E. / Terpos, E. / Filippakopoulos, P. / Muller, S. / Skaltsounis, A.L. / Downs, J.A. / Knapp, S. / Mikros, E. |
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手法 | X線回折 |
解像度 | 1.7 - 2.4 Å |
構造データ | ![]() PDB-5hrv: ![]() PDB-5hrw: ![]() PDB-5hrx: ![]() PDB-5ii1: ![]() PDB-5ii2: ![]() PDB-5iid: |
化合物 | ![]() ChemComp-64C: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-64E: ![]() ChemComp-SO4: ![]() ChemComp-64F: ![]() ChemComp-6BL: ![]() ChemComp-K: ![]() ChemComp-CIT: ![]() ChemComp-LU2: ![]() ChemComp-6BK: |
由来 |
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![]() | TRANSCRIPTION / BRM1 / BRG1-associated factor 180 / chromatin remodeling / PBRM1 / bromodomain / complex / small molecule / structural genomics consortium / SGC |