| タイトル | mTOR kinase structure, mechanism and regulation. |
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| ジャーナル・号・ページ | Nature, Vol. 497, Page 217-223, Year 2013 |
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| 掲載日 | 2013年3月22日 (構造データの登録日) |
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著者 | Yang, H. / Rudge, D.G. / Koos, J.D. / Vaidialingam, B. / Yang, H.J. / Pavletich, N.P. |
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リンク | Nature / PubMed:23636326 |
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| 手法 | X線回折 |
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| 解像度 | 3.2 - 3.6 Å |
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| 構造データ | PDB-4jsn: structure of mTORdeltaN-mLST8 complex 手法: X-RAY DIFFRACTION / 解像度: 3.2 Å PDB-4jsp: structure of mTORDeltaN-mLST8-ATPgammaS-Mg complex 手法: X-RAY DIFFRACTION / 解像度: 3.3 Å PDB-4jsv: mTOR kinase structure, mechanism and regulation. 手法: X-RAY DIFFRACTION / 解像度: 3.5 Å PDB-4jsx: structure of mTORDeltaN-mLST8-Torin2 complex 手法: X-RAY DIFFRACTION / 解像度: 3.5 Å PDB-4jt5: mTORdeltaN-mLST8-pp242 complex 手法: X-RAY DIFFRACTION / 解像度: 3.45 Å PDB-4jt6: structure of mTORDeltaN-mLST8-PI-103 complex 手法: X-RAY DIFFRACTION / 解像度: 3.6 Å |
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| 化合物 | ChemComp-AGS: PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER / ATP-gamma-S, エネルギー貯蔵分子類似体*YM
ChemComp-ADP: ADENOSINE-5'-DIPHOSPHATE / ADP, エネルギー貯蔵分子*YM
ChemComp-17G: 9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1H)-one
ChemComp-P2X: 2-[4-amino-1-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl]-1H-indol-5-ol
ChemComp-X6K: 3-(4-MORPHOLIN-4-YLPYRIDO[3',2':4,5]FURO[3,2-D]PYRIMIDIN-2-YL)PHENOL
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| 由来 | homo sapiens (ヒト)
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キーワード | TRANSFERASE / helical repeat / kinase / wd40 repeat / protein kinase / Raptor / transferase/transferase inhibitor / transferase-transferase inhibitor complex |
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