タイトル | A Combination of Spin Diffusion Methods for the Determination of Protein-Ligand Complex Structural Ensembles. |
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ジャーナル・号・ページ | Angew. Chem. Int. Ed. Engl., Vol. 54, Page 6511-, Year 2015 |
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掲載日 | 2013年9月9日 (構造データの登録日) |
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著者 | Pilger, J. / Mazur, A. / Monecke, P. / Schreuder, H. / Elshorst, B. / Bartoschek, S. / Langer, T. / Schiffer, A. / Krimm, I. / Wegstroth, M. ...Pilger, J. / Mazur, A. / Monecke, P. / Schreuder, H. / Elshorst, B. / Bartoschek, S. / Langer, T. / Schiffer, A. / Krimm, I. / Wegstroth, M. / Lee, D. / Hessler, G. / Wendt, K. / Becker, S. / Griesinger, C. |
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リンク | Angew. Chem. Int. Ed. Engl. / PubMed:25877959 |
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手法 | X線回折 |
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解像度 | 2 - 2.41 Å |
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構造データ | PDB-4c4x: Crystal structure of human bifunctional epoxide hydroxylase 2 complexed with C9 手法: X-RAY DIFFRACTION / 解像度: 2.17 Å PDB-4c4y: Crystal structure of human bifunctional epoxide hydroxylase 2 complexed with A4 手法: X-RAY DIFFRACTION / 解像度: 2.41 Å PDB-4c4z: Crystal structure of human bifunctional epoxide hydroxylase 2 complexed with A8 手法: X-RAY DIFFRACTION / 解像度: 2.06 Å PDB-4yxr: CRYSTAL STRUCTURE OF PKA IN COMPLEX WITH inhibitor. 手法: X-RAY DIFFRACTION / 解像度: 2.0 Å PDB-4yxs: CAMP-DEPENDENT PROTEIN KINASE PKA CATALYTIC SUBUNIT WITH PKI-5-24 手法: X-RAY DIFFRACTION / 解像度: 2.11 Å |
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化合物 | ChemComp-7WI: 1-(3-chlorophenyl)-3-(2-methoxyethyl)urea
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由来 | ![](img/tx_human.gif) homo sapiens (ヒト)![](img/tx_mammal.gif) ![](data/taxo/icon/Bos_taurus_S.png) bos taurus (ウシ)![](img/tx_mammal.gif) ![](data/taxo/icon/Oryctolagus_cuniculus_S.png) oryctolagus cuniculus (ウサギ)
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キーワード | HYDROLASE (加水分解酵素) / DRUG DESIGN (医薬品設計) / MULTIPLE BINDING MODES / TRANSFERASE (転移酵素) / COMPLEX (PHOSPHOTRANSFERASE-INHIBITOR) complex / TRANSFERASE/INHIBITOR / ATP-BINDING / PHOSPHOPROTEIN / SERINE/THREONINE-PROTEIN KINASE / CAMP (CAMP) / PROTEIN KINASE INHIBITOR / TRANSFERASE-IN COMPLEX / TRANSFERASE-INHIBITOR complex |
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