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-Structure paper
タイトル | Selectivity, Co-Crystal Structures and Neuroprotective Properties of Leucettines, a Family of Protein Kinase Inhibitors Derived from the Marine Sponge Alkaloid Leucettamine B. |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 55, Page 9312-, Year 2012 |
掲載日 | 2012年6月25日 (構造データの登録日) |
著者 | Tahtouh, T. / Elkins, J.M. / Filippakopoulos, P. / Soundararajan, M. / Burgy, G. / Durieu, E. / Cochet, C. / Schmid, R.S. / Lo, D.C. / Delhommel, F. ...Tahtouh, T. / Elkins, J.M. / Filippakopoulos, P. / Soundararajan, M. / Burgy, G. / Durieu, E. / Cochet, C. / Schmid, R.S. / Lo, D.C. / Delhommel, F. / Oberholzer, A. / Laurence, P. / Carreaux, F. / Bazureau, J.P. / Knapp, S. / Meijer, L. |
リンク | J. Med. Chem. / PubMed:22998443 |
手法 | X線回折 |
解像度 | 2 - 3.15 Å |
構造データ | PDB-4aze: PDB-4azf: PDB-4b7t: PDB-4gw8: |
化合物 | ChemComp-3RA: ChemComp-EDO: ChemComp-PO4: ChemComp-HOH: ChemComp-CWT: |
由来 |
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キーワード | TRANSFERASE / TRANSFERASE/PEPTIDE / TRANSFERASE-PEPTIDE COMPLEX / INSULIN PATHWAY / WNT SIGNALING PATHWAY / INHIBITOR / ONCOGENE / KINASE / SERINE-THREONINE / PIM1 / STRUCTURAL GENOMICS CONSORTIUM / SGC / ALTERNATIVE INITIATION / ATP-BINDING / MANGANESE / MEMBRANE / METAL-BINDING / NUCLEOTIDE-BINDING / NUCLEUS / PHOSPHOPROTEIN / PROTO-ONCOGENE / SERINE/THREONINE-PROTEIN KINASE / HOST-VIRUS INTERACTION / VIRAL IMMUNOEVASION / VIRION / VIRULENCE / CELL CYCLE / CELL MEMBRANE |