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-Structure paper
タイトル | Novel adenosine-derived inhibitors of 70 kDa heat shock protein, discovered through structure-based design |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 52, Page 1510-1513, Year 2009 |
掲載日 | 2009年1月26日 (構造データの登録日) |
![]() | Williamson, D.S. / Borgognoni, J. / Clay, A. / Daniels, Z. / Dokurno, P. / Drysdale, M.J. / Foloppe, N. / Francis, G.L. / Graham, C.J. / Howes, R. ...Williamson, D.S. / Borgognoni, J. / Clay, A. / Daniels, Z. / Dokurno, P. / Drysdale, M.J. / Foloppe, N. / Francis, G.L. / Graham, C.J. / Howes, R. / Macias, A.T. / Murray, J.B. / Parsons, R. / Shaw, T. / Surgenor, A.E. / Terry, L. / Wang, Y. / Wood, M. / Massey, A.J. |
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手法 | X線回折 |
解像度 | 2 - 2.3 Å |
構造データ | ![]() PDB-3fzf: ![]() PDB-3fzh: ![]() PDB-3fzk: ![]() PDB-3fzl: ![]() PDB-3fzm: |
化合物 | ![]() ChemComp-ATP: ![]() ChemComp-HOH: ![]() ChemComp-3BH: ![]() ChemComp-TRS: ![]() ChemComp-CL: ![]() ChemComp-3BK: ![]() ChemComp-3FD: ![]() ChemComp-3GO: |
由来 |
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![]() | CHAPERONE / HSP70 / HSC70 / BAG1 / heat shock / protein folding / adenosine / nucleoside / nucleotide exchange factor / small molecule inhibitor / ATP-binding / nucleotide-binding / stress response / apoptosis / nucleotide |