+Search query
-Structure paper
Title | Mechanism of small molecule inhibition of Plasmodium falciparum myosin A informs antimalarial drug design. |
---|---|
Journal, issue, pages | Nat Commun, Vol. 14, Page 3463-3463, Year 2023 |
Publish date | May 31, 2022 (structure data deposition date) |
Authors | Moussaoui, D. / Robblee, J.P. / Robert-Paganin, J. / Auguin, D. / Fisher, F. / Fagnant, P.M. / Macfarlane, J.E. / Schaletzky, J. / Wehri, E. / Mueller-Dieckmann, C. ...Moussaoui, D. / Robblee, J.P. / Robert-Paganin, J. / Auguin, D. / Fisher, F. / Fagnant, P.M. / Macfarlane, J.E. / Schaletzky, J. / Wehri, E. / Mueller-Dieckmann, C. / Baum, J. / Trybus, K.M. / Houdusse, A. |
External links | Nat Commun / PubMed:37308472 |
Methods | X-ray diffraction |
Resolution | 2.03 - 2.21 Å |
Structure data | PDB-8a12: PDB-8cdq: |
Chemicals | ChemComp-ADP: ChemComp-SO4: ChemComp-EDO: ChemComp-MG: ChemComp-HOH: ChemComp-GOL: ChemComp-PG4: ChemComp-AGS: ChemComp-KQ0: |
Source |
|
Keywords | MOTOR PROTEIN / Malaria / Plasmodium falciparum / Myosin A / Knx002 / antimalarial treatment / molecular motors / KNX-002 |