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-Structure paper
Title | Phenotypic Discovery of Triazolo[1,5- c ]quinazolines as a First-In-Class Bone Morphogenetic Protein Amplifier Chemotype. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 15263-15281, Year 2022 |
Publish date | Mar 24, 2021 (structure data deposition date) |
Authors | Wesseler, F. / Lohmann, S. / Riege, D. / Halver, J. / Roth, A. / Pichlo, C. / Weber, S. / Takamiya, M. / Muller, E. / Ketzel, J. ...Wesseler, F. / Lohmann, S. / Riege, D. / Halver, J. / Roth, A. / Pichlo, C. / Weber, S. / Takamiya, M. / Muller, E. / Ketzel, J. / Flegel, J. / Gihring, A. / Rastegar, S. / Bertrand, J. / Baumann, U. / Knippschild, U. / Peifer, C. / Sievers, S. / Waldmann, H. / Schade, D. |
External links | J. Med. Chem. / PubMed:36346705 |
Methods | X-ray diffraction |
Resolution | 1.85 Å |
Structure data | PDB-7nzy: |
Chemicals | ChemComp-UX2: ChemComp-MLI: ChemComp-PO4: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / Kinase / Inhibitor / Complex / ATP-competitive |