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-Structure paper
Title | Mining Public Domain Data to Develop Selective DYRK1A Inhibitors. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 11, Page 1620-1626, Year 2020 |
Publish date | Jun 18, 2019 (structure data deposition date) |
Authors | Henderson, S.H. / Sorrell, F. / Bennett, J. / Hanley, M.T. / Robinson, S. / Hopkins Navratilova, I. / Elkins, J.M. / Ward, S.E. |
External links | Acs Med. Chem. Lett. / PubMed:32832032 |
Methods | X-ray diffraction |
Resolution | 2.38 Å |
Structure data | PDB-6s1i: |
Chemicals | ChemComp-SO4: ChemComp-PG4: ChemComp-KR8: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / Kinase / catalytic domain / phosphorylated |