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-Structure paper
Title | Crystal Structure of the Human vaccinia-related kinase bound to a N,N-dipropynyl-dihydropteridine-3-hydroxyindazole inhibitor |
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Journal, issue, pages | To Be Published |
Publish date | Jan 18, 2019 (structure data deposition date) |
Authors | Counago, R.M. / dos Reis, C.V. / Takarada, J.E. / Azevedo, H. / Guimaraes, C. / Mascarello, A. / Gama, F. / Ferreira, M. / Massirer, K.B. / Arruda, P. ...Counago, R.M. / dos Reis, C.V. / Takarada, J.E. / Azevedo, H. / Guimaraes, C. / Mascarello, A. / Gama, F. / Ferreira, M. / Massirer, K.B. / Arruda, P. / Edwards, A.M. / Elkins, J.M. / Structural Genomics Consortium (SGC) |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | PDB-6npn: |
Chemicals | ChemComp-KWJ: ChemComp-SO4: ChemComp-EDO: ChemComp-PEG: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / transferase / protein kinase domain / Structural Genomics / Structural Genomics Consortium / SGC / Transferase-Transferase Inhibitor Complex |