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Title | New Irreversible alpha-l-Iduronidase Inhibitors and Activity-Based Probes. |
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Journal, issue, pages | Chemistry, Vol. 24, Page 19081-19088, Year 2018 |
Publish date | Nov 15, 2018 (structure data deposition date) |
Authors | Artola, M. / Kuo, C.L. / McMahon, S.A. / Oehler, V. / Hansen, T. / van der Lienden, M. / He, X. / van den Elst, H. / Florea, B.I. / Kermode, A.R. ...Artola, M. / Kuo, C.L. / McMahon, S.A. / Oehler, V. / Hansen, T. / van der Lienden, M. / He, X. / van den Elst, H. / Florea, B.I. / Kermode, A.R. / van der Marel, G.A. / Gloster, T.M. / Codee, J.D.C. / Overkleeft, H.S. / Aerts, J.M.F.G. |
External links | Chemistry / PubMed:30307091 |
Methods | X-ray diffraction |
Resolution | 2.02 - 2.39 Å |
Structure data | PDB-6i6r: PDB-6i6x: |
Chemicals | ChemComp-H62: ChemComp-NAG: ChemComp-GOL: ChemComp-TLA: ChemComp-CL: ChemComp-HOH: ChemComp-H6B: |
Source |
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Keywords | HYDROLASE / Iduronidase Inhibitors GH39 |