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Title | X-ray Structures and Feasibility Assessment of CLK2 Inhibitors for Phelan-McDermid Syndrome. |
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Journal, issue, pages | ChemMedChem, Vol. 13, Page 1997-2007, Year 2018 |
Publish date | Mar 12, 2018 (structure data deposition date) |
Authors | Kallen, J. / Bergsdorf, C. / Arnaud, B. / Bernhard, M. / Brichet, M. / Cobos-Correa, A. / Elhajouji, A. / Freuler, F. / Galimberti, I. / Guibourdenche, C. ...Kallen, J. / Bergsdorf, C. / Arnaud, B. / Bernhard, M. / Brichet, M. / Cobos-Correa, A. / Elhajouji, A. / Freuler, F. / Galimberti, I. / Guibourdenche, C. / Haenni, S. / Holzinger, S. / Hunziker, J. / Izaac, A. / Kaufmann, M. / Leder, L. / Martus, H.J. / von Matt, P. / Polyakov, V. / Roethlisberger, P. / Roma, G. / Stiefl, N. / Uteng, M. / Lerchner, A. |
External links | ChemMedChem / PubMed:29985556 |
Methods | X-ray diffraction |
Resolution | 1.42 - 2.6 Å |
Structure data | PDB-6fyi: PDB-6fyk: PDB-6fyl: PDB-6fyo: PDB-6fyp: PDB-6fyr: PDB-6fyv: |
Chemicals | ChemComp-EAE: ChemComp-HOH: ChemComp-EAZ: ChemComp-3NG: ChemComp-EAQ: ChemComp-SO4: |
Source |
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Keywords | TRANSFERASE / SPLICING / PHOSPHOTRANSFERASE / KINASE / TYROSINE-PROTEIN KINASE / SERINE/ THREONINE- PROTEIN KINASE / NUCLEOTIDE-BINDING |