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-Structure paper
Title | Design of KDM4 Inhibitors with Antiproliferative Effects in Cancer Models. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 8, Page 869-874, Year 2017 |
Publish date | Apr 11, 2017 (structure data deposition date) |
Authors | Chen, Y.K. / Bonaldi, T. / Cuomo, A. / Del Rosario, J.R. / Hosfield, D.J. / Kanouni, T. / Kao, S.C. / Lai, C. / Lobo, N.A. / Matuszkiewicz, J. ...Chen, Y.K. / Bonaldi, T. / Cuomo, A. / Del Rosario, J.R. / Hosfield, D.J. / Kanouni, T. / Kao, S.C. / Lai, C. / Lobo, N.A. / Matuszkiewicz, J. / McGeehan, A. / O'Connell, S.M. / Shi, L. / Stafford, J.A. / Stansfield, R.K. / Veal, J.M. / Weiss, M.S. / Yuen, N.Y. / Wallace, M.B. |
External links | ACS Med Chem Lett / PubMed:28835804 |
Methods | X-ray diffraction |
Resolution | 2.07 - 2.48 Å |
Structure data | PDB-5vgi: PDB-5vmp: |
Chemicals | ChemComp-NI: ChemComp-ZN: ChemComp-9DJ: ChemComp-HOH: ChemComp-9FJ: |
Source |
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Keywords | OXIDOREDUCTASE/INHIBITOR / KDM4 / Protein-Inhibitor Complex / demethylase / epigenetics / OXIDOREDUCTASE-INHIBITOR complex / Inhibitor-complex |