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-Structure paper
Title | Detection of Active Mammalian GH31 alpha-Glucosidases in Health and Disease Using In-Class, Broad-Spectrum Activity-Based Probes. |
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Journal, issue, pages | Acs Cent. Sci., Vol. 2, Page 351-358, Year 2016 |
Publish date | Feb 8, 2016 (structure data deposition date) |
Authors | Jiang, J. / Kuo, C.L. / Wu, L. / Franke, C. / Kallemeijn, W.W. / Florea, B.I. / van Meel, E. / van der Marel, G.A. / Codee, J.D. / Boot, R.G. ...Jiang, J. / Kuo, C.L. / Wu, L. / Franke, C. / Kallemeijn, W.W. / Florea, B.I. / van Meel, E. / van der Marel, G.A. / Codee, J.D. / Boot, R.G. / Davies, G.J. / Overkleeft, H.S. / Aerts, J.M. |
External links | Acs Cent. Sci. / PubMed:27280170 |
Methods | X-ray diffraction |
Resolution | 1.85 - 1.95 Å |
Structure data | PDB-5i23: PDB-5i24: |
Chemicals | ChemComp-PG4: ChemComp-SO4: ChemComp-EDO: ChemComp-66V: ChemComp-HOH: ChemComp-66U: ChemComp-TRS: |
Source |
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Keywords | TRANSFERASE / Alpha glycosidase / Cyclophellitol Aziridine / Inhibitor / Probe / HYDROLASE |