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Title | Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 6844-6863, Year 2015 |
Publish date | Aug 3, 2015 (structure data deposition date) |
![]() | Engel, J. / Richters, A. / Getlik, M. / Tomassi, S. / Keul, M. / Termathe, M. / Lategahn, J. / Becker, C. / Mayer-Wrangowski, S. / Grutter, C. ...Engel, J. / Richters, A. / Getlik, M. / Tomassi, S. / Keul, M. / Termathe, M. / Lategahn, J. / Becker, C. / Mayer-Wrangowski, S. / Grutter, C. / Uhlenbrock, N. / Krull, J. / Schaumann, N. / Eppmann, S. / Kibies, P. / Hoffgaard, F. / Heil, J. / Menninger, S. / Ortiz-Cuaran, S. / Heuckmann, J.M. / Tinnefeld, V. / Zahedi, R.P. / Sos, M.L. / Schultz-Fademrecht, C. / Thomas, R.K. / Kast, S.M. / Rauh, D. |
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Methods | X-ray diffraction |
Resolution | 2.3 - 3 Å |
Structure data | ![]() PDB-5d10: ![]() PDB-5d11: ![]() PDB-5d12: |
Chemicals | ![]() ChemComp-563: ![]() ChemComp-HOH: ![]() ChemComp-GOL: ![]() ChemComp-56G: ![]() ChemComp-G97: |
Source |
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![]() | TRANSFERASE / kinase inhibitor / drug resistance |