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-Structure paper
Title | Thiophenecarboxamide Derivatives Activated by EthA Kill Mycobacterium tuberculosis by Inhibiting the CTP Synthetase PyrG. |
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Journal, issue, pages | Chem. Biol., Vol. 22, Page 917-927, Year 2015 |
Publish date | Apr 17, 2015 (structure data deposition date) |
![]() | Mori, G. / Chiarelli, L.R. / Esposito, M. / Makarov, V. / Bellinzoni, M. / Hartkoorn, R.C. / Degiacomi, G. / Boldrin, F. / Ekins, S. / de Jesus Lopes Ribeiro, A.L. ...Mori, G. / Chiarelli, L.R. / Esposito, M. / Makarov, V. / Bellinzoni, M. / Hartkoorn, R.C. / Degiacomi, G. / Boldrin, F. / Ekins, S. / de Jesus Lopes Ribeiro, A.L. / Marino, L.B. / Centarova, I. / Svetlikova, Z. / Blasko, J. / Kazakova, E. / Lepioshkin, A. / Barilone, N. / Zanoni, G. / Porta, A. / Fondi, M. / Fani, R. / Baulard, A.R. / Mikusova, K. / Alzari, P.M. / Manganelli, R. / de Carvalho, L.P. / Riccardi, G. / Cole, S.T. / Pasca, M.R. |
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Methods | X-ray diffraction |
Resolution | 1.99 - 3.52 Å |
Structure data | ![]() PDB-4zdi: ![]() PDB-4zdj: ![]() PDB-4zdk: |
Chemicals | ![]() ChemComp-CA: ![]() ChemComp-UTP: ![]() ChemComp-MG: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-ONL: ![]() ChemComp-ACP: |
Source |
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![]() | LIGASE / CTP synthase / PyrG / amidotransferase / UTP / AMP-PCP / 5-oxo-L-norleucine |