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-Structure paper
Title | Isoform-Selective and Stereoselective Inhibition of Hypoxia Inducible Factor-2. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 5930-5941, Year 2015 |
Publish date | Jan 22, 2015 (structure data deposition date) |
![]() | Scheuermann, T.H. / Stroud, D. / Sleet, C.E. / Bayeh, L. / Shokri, C. / Wang, H. / Caldwell, C.G. / Longgood, J. / MacMillan, J.B. / Bruick, R.K. ...Scheuermann, T.H. / Stroud, D. / Sleet, C.E. / Bayeh, L. / Shokri, C. / Wang, H. / Caldwell, C.G. / Longgood, J. / MacMillan, J.B. / Bruick, R.K. / Gardner, K.H. / Tambar, U.K. |
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Methods | X-ray diffraction |
Resolution | 1.698 Å |
Structure data | ![]() PDB-4xt2: |
Chemicals | ![]() ChemComp-43L: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / transcription factor / Hypoxia Inducible Factor / inhibitor / cancer |