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-Structure paper
Title | A small-molecule mimic of a peptide docking motif inhibits the protein kinase PDK1. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. USA, Vol. 111, Page 18590-18595, Year 2014 |
Publish date | Nov 3, 2014 (structure data deposition date) |
![]() | Rettenmaier, T.J. / Sadowsky, J.D. / Thomsen, N.D. / Chen, S.C. / Doak, A.K. / Arkin, M.R. / Wells, J.A. |
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Methods | X-ray diffraction |
Resolution | 1.412 - 1.55 Å |
Structure data | ![]() PDB-4rqk: ![]() PDB-4rqv: ![]() PDB-4rrv: |
Chemicals | ![]() ChemComp-GOL: ![]() ChemComp-ATP: ![]() ChemComp-R1S: ![]() ChemComp-EPE: ![]() ChemComp-HOH: ![]() ChemComp-R2S: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Protein Kinase / Phosphorylation / TRANSFERASE-TRANSFERASE INHIBITOR complex / PIFtide |