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-Structure paper
Title | Discovery and Optimization of a Novel Series of Potent Mutant B-Raf V600E Selective Kinase Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 56, Page 1996-, Year 2013 |
Publish date | Sep 19, 2012 (structure data deposition date) |
![]() | Vasbinder, M.M. / Aquila, B. / Augustin, M. / Chen, H. / Cheung, T. / Cook, D. / Drew, L. / Fauber, B.P. / Glossop, S. / Grondine, M. ...Vasbinder, M.M. / Aquila, B. / Augustin, M. / Chen, H. / Cheung, T. / Cook, D. / Drew, L. / Fauber, B.P. / Glossop, S. / Grondine, M. / Hennessy, E.J. / Johannes, J. / Lee, S. / Lyne, P.D. / Mortl, M. / Omer, C. / Palakurthi, S. / Pontz, T. / Read, J. / Sha, L. / Shen, M. / Steinbacher, S. / Wang, H. / Wu, A. / Ye, M. |
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Methods | X-ray diffraction |
Resolution | 1.65 - 3.1 Å |
Structure data | ![]() PDB-4bb4: ![]() PDB-4h58: |
Chemicals | ![]() ChemComp-32W: ![]() ChemComp-MG: ![]() ChemComp-HOH: ![]() ChemComp-10Z: ![]() ChemComp-CL: |
Source |
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![]() | TRANSFERASE / UNPHOSPHORYLATED / TRANSFERASE/TRANSFERASE INHIBITOR / protein kinase / structure based drug discovery / TRANSFERASE-TRANSFERASE INHIBITOR complex |