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-Structure paper
Title | The Discovery of a Novel Series of Potent and Orally Bioavailable Phosphoinositide 3-Kinase Gamma Inhibitors |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 5467-, Year 2012 |
Publish date | Mar 22, 2012 (structure data deposition date) |
Authors | Leahy, J.W. / Buhr, C.A. / Johnson, H.W.B. / Kim, B.G. / Baik, T. / Cannoy, J. / Forsyth, T.P. / Jeong, J.W. / Lee, M.S. / Ma, S. ...Leahy, J.W. / Buhr, C.A. / Johnson, H.W.B. / Kim, B.G. / Baik, T. / Cannoy, J. / Forsyth, T.P. / Jeong, J.W. / Lee, M.S. / Ma, S. / Noson, K. / Wang, L. / Williams, M. / Nuss, J.M. / Brooks, E. / Heald, N. / Holst, C. / Jaeger, C. / Lam, S. / Lougheed, J.C. / Nguyen, L. / Plonowski, A. / Stout, T. / Foster, P.G. / Wu, X. / Yakes, M.F. / Yu, R. / Zhang, W. / Lamb, P. / Raeber, O. |
External links | J. Med. Chem. / PubMed:22548342 |
Methods | X-ray diffraction |
Resolution | 2.13 - 2.81 Å |
Structure data | PDB-4anu: PDB-4anv: PDB-4anw: PDB-4anx: |
Chemicals | ChemComp-SO4: ChemComp-EM7: ChemComp-HOH: ChemComp-751: ChemComp-O92: ChemComp-534: |
Source |
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Keywords | TRANSFERASE |