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-Structure paper
Title | Structural Analysis of the Mechanism of Inhibition and Allosteric Activation of the Kinase Domain of HER2 Protein. |
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Journal, issue, pages | J. Biol. Chem., Vol. 286, Page 18756-18765, Year 2011 |
Publish date | Nov 23, 2010 (structure data deposition date) |
![]() | Aertgeerts, K. / Skene, R. / Yano, J. / Sang, B.C. / Zou, H. / Snell, G. / Jennings, A. / Iwamoto, K. / Habuka, N. / Hirokawa, A. ...Aertgeerts, K. / Skene, R. / Yano, J. / Sang, B.C. / Zou, H. / Snell, G. / Jennings, A. / Iwamoto, K. / Habuka, N. / Hirokawa, A. / Ishikawa, T. / Tanaka, T. / Miki, H. / Ohta, Y. / Sogabe, S. |
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Methods | X-ray diffraction |
Resolution | 1.5 - 2.25 Å |
Structure data | ![]() PDB-3poz: ![]() PDB-3pp0: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-03P: ![]() ChemComp-HOH: ![]() ChemComp-03Q: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / KINASE DOMAIN / ANTI-ONCOGENE / ATP-BINDING / CELL CYCLE / DISEASE MUTATION / GLYCOPROTEIN / MEMBRANE / NUCLEOTIDE-BINDING / PHOSPHOPROTEIN / RECEPTOR / SECRETED / TRANSFERASE / TRANSMEMBRANE / TYROSINE-PROTEIN KINASE / TRANSFERASE-TRANSFERASE INHIBITOR complex / TYROSINE KINASE INHIBITOR |