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-Structure paper
Title | Halogen bonds form the basis for selective P-TEFb inhibition by DRB |
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Journal, issue, pages | Chem. Biol., Vol. 17, Page 931-936, Year 2010 |
Publish date | May 9, 2010 (structure data deposition date) |
Authors | Baumli, S. / Endicott, J.A. / Johnson, L.N. |
External links | Chem. Biol. / PubMed:20851342 |
Methods | X-ray diffraction |
Resolution | 2.1 - 2.8 Å |
Structure data | PDB-3my1: PDB-3my5: |
Chemicals | ChemComp-PO4: ChemComp-GOL: ChemComp-RFZ: ChemComp-HOH: ChemComp-FMT: ChemComp-SGM: |
Source |
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Keywords | TRANSCRIPTION/PROTEIN BINDING/INHIBITOR / CDK-cyclin complex / phosphorylated / TRANSCRIPTION-PROTEIN BINDING-INHIBITOR complex / TRANSFERASE/PROTEIN BINDING/INHIBITOR / CDK / cyclin / inhibitor / DRB / TRANSFERASE-PROTEIN BINDING-INHIBITOR complex |