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-Structure paper
Title | Binding thermodynamics of substituted diaminopyrimidine renin inhibitors. |
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Journal, issue, pages | Anal. Biochem., Vol. 360, Page 30-40, Year 2007 |
Publish date | Oct 2, 2006 (structure data deposition date) |
Authors | Sarver, R.W. / Peevers, J. / Cody, W.L. / Ciske, F.L. / Dyer, J. / Emerson, S.D. / Hagadorn, J.C. / Holsworth, D.D. / Jalaie, M. / Kaufman, M. ...Sarver, R.W. / Peevers, J. / Cody, W.L. / Ciske, F.L. / Dyer, J. / Emerson, S.D. / Hagadorn, J.C. / Holsworth, D.D. / Jalaie, M. / Kaufman, M. / Mastronardi, M. / McConnell, P. / Powell, N.A. / Quin, J. / Van Huis, C.A. / Zhang, E. / Mochalkin, I. |
External links | Anal. Biochem. / PubMed:17113558 |
Methods | X-ray diffraction |
Resolution | 1.9 - 2.6 Å |
Structure data | PDB-2iko: PDB-2iku: PDB-2il2: |
Chemicals | ChemComp-7IG: ChemComp-HOH: ChemComp-LIY: ChemComp-LIX: ChemComp-CIT: |
Source |
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Keywords | HYDROLASE / Renin / Inhibitors / Drug Design |