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Title | High Resolution Crystal Structures of HIV-1 Protease with a Potent Non-Peptide Inhibitor (Uic-94017) Active Against Multi-Drug-Resistant Clinical Strains. |
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Journal, issue, pages | J. Mol. Biol., Vol. 338, Page 341-352, Year 2004 |
Publish date | Sep 15, 2006 (structure data deposition date) |
![]() | Tie, Y. / Boross, P.I. / Wang, Y.F. / Gaddis, L. / Hussain, A.K. / Leshchenko, S. / Ghosh, A.K. / Louis, J.M. / Harrison, R.W. / Weber, I.T. |
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Methods | X-ray diffraction |
Resolution | 1.1 - 1.53 Å |
Structure data | ![]() PDB-2idw: ![]() PDB-2ien: ![]() PDB-2ieo: |
Chemicals | ![]() ChemComp-CL: ![]() ChemComp-PO4: ![]() ChemComp-DMS: ![]() ChemComp-ACY: ![]() ChemComp-GOL: ![]() ChemComp-017: ![]() ChemComp-HOH: ![]() ChemComp-NA: |
Source |
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![]() | HYDROLASE / HIV-1 PROTEASE / MUTANT / DIMER / INHIBITOR / UIC-94017 / TMC114 / darunavir / I84V |